021-51111890
购物车（）
sales@molnova.cn
Asenapine maleate
CAS No. 85650-56-2
Asenapine maleate ( Org 5222 maleate;Org-5222 maleate;Org5222 maleate )
产品货号. M16209 CAS No. 85650-56-2
Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥243 | 有现货 |
|
| 10MG | ￥381 | 有现货 |
|
| 25MG | ￥591 | 有现货 |
|
| 50MG | ￥786 | 有现货 |
|
| 100MG | ￥1110 | 有现货 |
|
| 200MG | ￥1920 | 有现货 |
|
| 500MG | ￥3175 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称Asenapine maleate
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
-
产品描述Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors; shows much lower affinity (pKi<5) for muscarinic receptor; behaves as a potent antagonist 5-HT receptors (5-HT2A pKB=9.0), dopaime and adrenoceptors; shows strong antipsychotic potential in vivo.Schizophrenia Approved
-
同义词Org 5222 maleate;Org-5222 maleate;Org5222 maleate
-
通路Angiogenesis
-
靶点Adrenergic Receptor
-
受体5-HT2A;5-HT2B;5-HT2C;5-HT6;5-HT7
-
研究领域Neurological Disease
-
适应症Schizophrenia
化学信息
-
CAS Number85650-56-2
-
分子量401.84
-
分子式C21H20ClNO5
-
纯度>98% (HPLC)
-
溶解度10 mM in DMSO
-
SMILESCN1C[C@H]2[C@H](C1)C3=C(C=CC(=C3)Cl)OC4=CC=CC=C24.C(=C\C(=O)O)\C(=O)O
-
化学全称1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1)
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1. Room P, et al. Eur J Pharmacol. 1991 Dec 3;205(3):233-40.
2. Broekkamp CL, et al. Arzneimittelforschung. 1990 May;40(5):544-9.
3. Psychopharmacology (Berl). 2008 Feb;196(3):417-29.
4. Shahid M, et al. J Psychopharmacol. 2009 Jan;23(1):65-73.
2. Broekkamp CL, et al. Arzneimittelforschung. 1990 May;40(5):544-9.
3. Psychopharmacology (Berl). 2008 Feb;196(3):417-29.
4. Shahid M, et al. J Psychopharmacol. 2009 Jan;23(1):65-73.
产品手册
关联产品
-
Naringenin chalcone
Naringenin chalcone has antiallergic activity .Naringenin chalcone suppresses asthmatic symptoms by inhibiting Th2 cytokine production from CD4 T cells.
-
Pimavanserin tartrat...
Pimavanserin is an effective and specific serotonin 5-HT2A inverse agonist (pIC50: 8.73), used in the therapy of psychosis associated with Parkinson’s disease.
-
DL-Adrenaline Hydroc...
The active sympathomimetic hormone from the adrenal medulla in most species.
